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Found 6 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] B' and Ligand = 'BDBM50018671'
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50018671(CHEMBL3291019)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of MAO-B in rat liver homogenate preincubated for 240 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50018671(CHEMBL3291019)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of MAO-B in rat liver homogenate preincubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50018671(CHEMBL3291019)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of MAO-B in rat liver homogenate preincubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50018671(CHEMBL3291019)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of MAO-B in rat liver homogenate using [14C]-phenylethylamine as substrate preincubated for 30 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50018671(CHEMBL3291019)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of human recombinant MAOB using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50018671(CHEMBL3291019)
Affinity DataIC50:  6.17E+4nMAssay Description:Inhibition of MAO-B in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed