Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity against GST-hARLBD was measured in SC-3 cell by using [3H]-testosterone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 154nMAssay Description:Inhibition of [3H]-Mibolerone binding to human Androgen receptor of PC3/AR Cell LysateMore data for this Ligand-Target Pair
Affinity DataIC50: 154nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human androgen receptor expressed in mouse NIH3T3 cells assessed as inhibition of DHT-induced transcriptional activation after...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at AR in human MDA-kb2 cells cotransfected with MMTV-luc assessed as decrease in DHT-induced luciferase activity by reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Antagonist activity at wild type human recombinant androgen receptor assessed as inhibition of testosterone-induced growth of mouse androgen dependen...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Antagonist activity at human androgen receptor expressed in human CV1 cells assessed as inhibition of receptor-mediated transactivation by MMTV-lucif...More data for this Ligand-Target Pair