Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) with Target = 'Aurora kinase A' and Ligand = 'BDBM87049'
TargetAurora kinase A(Human)
Moffitt Cancer Center

LigandPNGBDBM87049(Bisanilinopyrimidine inhibitor, 3)
Affinity DataIC50: 149nM Kd:  299nMpH: 7.4 T: 2°CAssay Description:The formation of ADP from ATP was quantified using a coupled enzyme assay (DiscoverX) in with a fluorescent resorufin dye is generated from the inter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2012
Entry Details Article
PubMed