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Found 4 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50355083'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataKi:  6.37E+3nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataKi:  6.37E+3nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataIC50:  3.41E+3nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataIC50: >6.47E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed