Affinity DataKi: 0.0650nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity against rat Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]Bradykinin from human recombinant bradykinin B2 receptor expressed in CHEM1 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]Bradykinin from human recombinant bradykinin B2 receptor expressed in CHEM1 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0490nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair