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Found 4 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor' and Ligand = 'BDBM50121684'
TargetB2 bradykinin receptor(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50121684(CHEMBL3616944)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]BK from B2R in guinea pig ileum membranes by liquid scintillation counting in based radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50121684(CHEMBL3616944)
Affinity DataKi:  1nMAssay Description:Binding affinity to B2R in guinea pig ileum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50121684(CHEMBL3616944)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [3H]BK from human B2R expressed in HEK293 cell membranes by liquid scintillation counting in based radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50121684(CHEMBL3616944)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]BK from B2R in rat brain membranes by liquid scintillation counting in based radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed