Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 0.0631nMAssay Description:Antagonist activity at guinea pig bradykinin B2 receptor in longitudinal smooth muscle assessed as inhibition of bradykinin-induced contractile respo...More data for this Ligand-Target Pair
Affinity DataKd: 0.316nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair