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Found 3 Enz. Inhib. hit(s) with Target = 'Beta-1/Beta-2/Beta-3 adrenergic receptor' and Ligand = 'BDBM50212981'
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataIC50:  0.900nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colon in presence of phentolamine (10 uM), desmethylimipramine (0.5 uM) and hydrocortisone (30 uM)More data for this Ligand-Target Pair
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TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataIC50:  480nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
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TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails