Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Beta-1/Beta-2/Beta-3 adrenergic receptor' and Ligand = 'BDBM50226717'
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50226717((+/-)-Pindobind | CHEMBL157881)
Affinity DataKi:  0.460nMAssay Description:In vitro inhibition against purified human erythrocyte carbonic anhydrase II was determined (acetozolamide used as control.)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50226717((+/-)-Pindobind | CHEMBL157881)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50226717((+/-)-Pindobind | CHEMBL157881)
Affinity DataKd:  2.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50226717((+/-)-Pindobind | CHEMBL157881)
Affinity DataKd:  1.60nMAssay Description:In vitro inhibition against purified human erythrocyte carbonic anhydrase II was determined (acetozolamide used as control.)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed