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Found 4 Enz. Inhib. hit(s) with Target = 'Beta-2 adrenergic receptor' and Ligand = 'BDBM50156304'
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156304(3-benzenesulfonyl-4-ethoxy-furazan 2-oxide | 4-eth...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156304(3-benzenesulfonyl-4-ethoxy-furazan 2-oxide | 4-eth...)
Affinity DataEC50:  1.20E+3nMAssay Description:Vasodilating activity against phenylephrine-induced contraction in rat thoracic aorta in presence of 1H-[1,2,4]oxadiazolo-[4,3-a]quinoxalin-1-oneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156304(3-benzenesulfonyl-4-ethoxy-furazan 2-oxide | 4-eth...)
Affinity DataEC50:  12nMAssay Description:Vasodilating activity against phenylephrine-induced contractions in rat thoracic aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156304(3-benzenesulfonyl-4-ethoxy-furazan 2-oxide | 4-eth...)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in prese...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed