Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Bile acid receptor' and Ligand = 'BDBM50258109'
TargetBile acid receptor(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50258109(CHEMBL4077016)
Affinity DataEC50:  0.300nMAssay Description:Transactivation of human FXR expressed in human HeLa cells co-expressing BSEP after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBile acid receptor(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50258109(CHEMBL4077016)
Affinity DataKd:  37nMAssay Description:Binding affinity to FXR (unknown origin) ligand binding domain by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed