Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3' and Ligand = 'BDBM50394617'
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataEC50:  58nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataIC50: 1.72nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed