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Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50260090'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50260090(CHEMBL4076296)
Affinity DataIC50:  27nMAssay Description:Inhibition of GST-tagged BRD4 (unknown origin) using biotinylated acetyl-histone H4 peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50260090(CHEMBL4076296)
Affinity DataIC50:  44nMAssay Description:Inhibition of recombinant GST-tagged BRD4 BD1 (44 to 168 residues) (unknown origin) incubated for 30 mins by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed