Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 3' and Ligand = 'BDBM50320127'
TargetC-X-C chemokine receptor type 3(Human)
Merck Serono

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320127BDBM50320127(N-(3-(1-(2-(4-((N-benzyl-4-chlorophenylsulfonamido...)
Affinity DataKi:  211nMAssay Description:Displacement of labeled ITAC from CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Merck Serono

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320127BDBM50320127(N-(3-(1-(2-(4-((N-benzyl-4-chlorophenylsulfonamido...)
Affinity DataKi:  348nMAssay Description:Displacement of labeled IP10 from CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Merck Serono

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320127BDBM50320127(N-(3-(1-(2-(4-((N-benzyl-4-chlorophenylsulfonamido...)
Affinity DataIC50: 538nMAssay Description:Antagonist activity at human CXCR3 expressed in mouse L1.2 cells assessed as inhibition of IP10-induced chemotaxis after 4 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Merck Serono

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320127BDBM50320127(N-(3-(1-(2-(4-((N-benzyl-4-chlorophenylsulfonamido...)
Affinity DataKi:  6.50E+3nMAssay Description:Antagonist activity at CXCR3 (unknown origin) assessed as reduction in CXCL10 induced calcium flux by FLIPR methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed