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Found 1 Enz. Inhib. hit(s) with Target = 'Calcitonin gene-related peptide 2' and Ligand = 'BDBM50570407'
TargetCalcitonin gene-related peptide 2(Homo sapiens)
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570407(CHEMBL4865654)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed