Affinity DataKi: 2.84E+3nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic & Petroleum Chemistry
Curated by ChEMBL
Institute Of Bioorganic & Petroleum Chemistry
Curated by ChEMBL
Affinity DataKi: 1.82E+7nMAssay Description:Binding affinity at cannabinoid receptor 1 using rat brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic & Petroleum Chemistry
Curated by ChEMBL
Institute Of Bioorganic & Petroleum Chemistry
Curated by ChEMBL
Affinity DataKi: 1.82E+7nMAssay Description:Cannabinoid receptor 1 binding affinity by measuring its ability to displace [3H]WIN-55212-2 in rat forebrain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic & Petroleum Chemistry
Curated by ChEMBL
Institute Of Bioorganic & Petroleum Chemistry
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Concentration of compound required to inhibit 50% of [3H]-WIN- 55212 binding to Cannabinoid receptor 1 in rat cerebellum membranes.More data for this Ligand-Target Pair