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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50310000'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50310000(4-((1H-1,2,4-Triazol-1-yl)methyl)-5-(4-bromophenyl...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50310000(4-((1H-1,2,4-Triazol-1-yl)methyl)-5-(4-bromophenyl...)
Affinity DataIC50:  2.51nMAssay Description:Inverse agonist activity at human recombinant CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed