Affinity DataKi: 13.3nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
Affinity DataKi: 13.8nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 35nM EC50: 798nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro inhibitory activity towards human cannabinoid receptors 2 using fluorescence assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataEC50: 30nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 634nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in HEK293 cells coexpressing Galphaq/o5 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair