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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50465029'
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Otago

Curated by ChEMBL
LigandPNGBDBM50465029(CHEMBL4283967)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Otago

Curated by ChEMBL
LigandPNGBDBM50465029(CHEMBL4283967)
Affinity DataIC50: >1.00E+4nMAssay Description:Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed