Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Carbonic anhydrase 9' and Ligand = 'BDBM50163861'
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163861(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKoff:  1.80E+6s-1Assay Description:Binding affinity to human recombinant CA9 catalytic domain assessed as association rate constant after 30 secs by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163861(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKd:  22nMAssay Description:Binding affinity to human recombinant CA9 catalytic domain by fluorescence-based thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163861(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.260M-1s-1Assay Description:Binding affinity to human recombinant CA9 catalytic domain assessed as dissociation rate constant after 30 secs by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163861(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKd:  150nMAssay Description:Binding affinity to human recombinant CA9 catalytic domain after 30 secs by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163861(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to human CA9 catalytic domain expressed in mammalian expression system assessed as intrinsic thermodynamic equilibrium constant at p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163861(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.260M-1s-1Assay Description:Binding affinity to human CA9 catalytic domain expressed in mammalian expression system assessed as dissociation rate constant at pH 7 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2019
Entry Details Article
PubMed