Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 1 Enz. Inhib. hit(s) with Target = 'Caspase-3' and Ligand = 'BDBM10297'
TargetCaspase-3(Human)
Glaxosmithkline

LigandPNGBDBM10297(1-methyl-5-nitro-2,3-dihydro-1H-indole-2,3-dione |...)
Affinity DataKi:  500nM ΔG°:  -36.6kJ/mole IC50:  1.00E+3nMpH: 7.5 T: 30°CAssay Description:The substrate peptides terminating in AMC/AFC are processed by caspases with or without inhibitors, and the accumulation of AMC/AFC was assessed with...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed