Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) with Target = 'Caspase-3' and Ligand = 'BDBM231'
TargetCaspase-3(Human)
Sunesis Pharmaceuticals

LigandPNGBDBM231(Heterocyclic deriv. 65a | 5-{[(3-{[(2S)-1-carboxy-...)
Affinity DataKi:  160nM ΔG°:  -38.8kJ/molepH: 7.4 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2003
Entry Details Article
PubMed