Found 3 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50016425'
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Mus musculus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.191nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair