Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50360276'
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-SR-27897 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed