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Found 2 Enz. Inhib. hit(s) with Target = 'Cruzipain' and Ligand = 'BDBM50306592'
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306592(3-(4-((S)-3-methyl-2-(quinolin-6-ylmethylamino)but...)
Affinity DataKi:  460nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306592(3-(4-((S)-3-methyl-2-(quinolin-6-ylmethylamino)but...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed