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Compile Data Set for Download or QSAR
maximum 50k data
Found
1
Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 12' and Ligand = 'BDBM2579'
Target
Cyclin-dependent kinase 12
(Homo sapiens)
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM2579
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
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Affinity Data
IC50: 53nM
Assay Description:
Inhibition of N-terminal FLAG-tagged human full-length CDK12 (1 to 1490 residues)/N-terminal His-tagged CycK (1 to 580 residues) expressed in Sf9 cel...
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