Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 2' and Ligand = 'BDBM50033098'
TargetCysteinyl leukotriene receptor 2(Human)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50033098(CHEMBL3342944)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at human CysLT2 expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization preincubated for 30 mins pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50033098(CHEMBL3342944)
Affinity DataIC50: 38nMAssay Description:Antagonist activity against CysLT2 receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of LTD4-induced calcium mobilization pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Setsunan University

Curated by ChEMBL
LigandPNGBDBM50033098(CHEMBL3342944)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed