Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 2D4' and Ligand = 'BDBM50122613'
TargetCytochrome P450 2D4(Rattus norvegicus)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50122613(3,4-dihydroisoquinoline-2(1H)-carboximidamide | CH...)
Affinity DataIC50:  7.47E+5nMAssay Description:Inhibition of MAMC O-dealkylation mediated by rat Cytochrome P450 2D4 expressed in Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed