Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM50620534'
TargetD(1A) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50620534BDBM50620534(CHEMBL5435602)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]SCH-23390 from human dopamine D1 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetD(1A) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50620534BDBM50620534(CHEMBL5435602)
Affinity DataIC50: 107nMAssay Description:Antagonist activity at human dopamine D1 receptor expressed in HEK-T cells assessed as inhibition of dopamine-induced cAMP production incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetD(1A) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50620534BDBM50620534(CHEMBL5435602)
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at N-terminal Flag epitope tagged human dopamine D1 receptor expressed in HTLA cells assessed as inhibition of dopamine-induced b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetD(1A) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50620534BDBM50620534(CHEMBL5435602)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human dopamine D1 receptor expressed in HEK-T cells assessed as cAMP production incubated for 15 mins by luciferase based Glosens...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetD(1A) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50620534BDBM50620534(CHEMBL5435602)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at N-terminal Flag epitope tagged human dopamine D1 receptor expressed in HTLA cells assessed as beta-arrestin translocation activit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed