Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50004921'
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004921BDBM50004921(CHEMBL34095 | (R)-3-Allyl-6-bromo-7,8-dihydroxy-1-...)
Affinity DataKd:  300nMAssay Description:In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Texas At Austin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004921BDBM50004921(CHEMBL34095 | (R)-3-Allyl-6-bromo-7,8-dihydroxy-1-...)
Affinity DataKi:  350nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004921BDBM50004921(CHEMBL34095 | (R)-3-Allyl-6-bromo-7,8-dihydroxy-1-...)
Affinity DataKd:  480nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004921BDBM50004921(CHEMBL34095 | (R)-3-Allyl-6-bromo-7,8-dihydroxy-1-...)
Affinity DataKd:  500nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004921BDBM50004921(CHEMBL34095 | (R)-3-Allyl-6-bromo-7,8-dihydroxy-1-...)
Affinity DataIC50: 511nMAssay Description:Displacement of [3H]YM-09151-2 (60 pm) from dopamine receptor D2 in crude membrane fraction of rat brain corpus striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004921BDBM50004921(CHEMBL34095 | (R)-3-Allyl-6-bromo-7,8-dihydroxy-1-...)
Affinity DataKd:  1.60E+3nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed