Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50007517'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Astra Research Centre

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataKi:  0.0640nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Astra Research Centre

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataKi:  0.0640nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Astra Research Centre

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal dopamine receptor D2 was determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Astra Research Centre

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataIC50:  1.40nMAssay Description:The affinity for the Dopamine receptor D2 was assessed by the inhibition of [3H]-spiperone binding in rat striatal membranes in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Astra Research Centre

Curated by ChEMBL
LigandPNGBDBM50007517((S)-3-bromo-N-((1-ethylpyrrolidin-2-yl)methyl)-2-h...)
Affinity DataIC50:  1.40nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed