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Found 2 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50021796'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021796(CHEMBL3299094)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021796(CHEMBL3299094)
Affinity DataEC50:  0.390nMAssay Description:Partial agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed