Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50091033'
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091033BDBM50091033(9-Carbamoyl-7-methyl-4,6,6a,7,8,9-hexahydro-indolo...)
Affinity DataKd:  0.620nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091033BDBM50091033(9-Carbamoyl-7-methyl-4,6,6a,7,8,9-hexahydro-indolo...)
Affinity DataKd:  1nMAssay Description:In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091033BDBM50091033(9-Carbamoyl-7-methyl-4,6,6a,7,8,9-hexahydro-indolo...)
Affinity DataKd:  1.80nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091033BDBM50091033(9-Carbamoyl-7-methyl-4,6,6a,7,8,9-hexahydro-indolo...)
Affinity DataKd:  2.80nMAssay Description:In vitro affinity at mutant D2 receptor (S193A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Texas

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50091033BDBM50091033(9-Carbamoyl-7-methyl-4,6,6a,7,8,9-hexahydro-indolo...)
Affinity DataKd:  2.80nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50091033BDBM50091033(9-Carbamoyl-7-methyl-4,6,6a,7,8,9-hexahydro-indolo...)
Affinity DataKi:  390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2011
Entry Details
PubMed