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Report error Found 11 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50252513'
TargetD(2) dopamine receptor(Human)
Acadia Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Acadia Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to D2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Acadia Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  2.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetD(2) dopamine receptor(Rat)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetD(2) dopamine receptor(Rat)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Acadia Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Acadia Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  4.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  6.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Acadia Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) after 60 mins by Ultra lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed