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Found 2 Enz. Inhib. hit(s) with Target = 'DNA gyrase subunit A' and Ligand = 'BDBM50178917'
TargetDNA gyrase subunit A(Staphylococcus aureus)
Achillion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50178917((S,Z)-7-(3-(aminomethyl)-4-(methoxyimino)pyrrolidi...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase Ser84Leu mutant assessed as inhibition of supercoiling of pBR322 DNA after 60 min by gel electrophores...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Staphylococcus aureus)
Achillion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50178917((S,Z)-7-(3-(aminomethyl)-4-(methoxyimino)pyrrolidi...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase gyrA S84L mutant supercoiling activity assessed as effect on conversion of relaxed pBR322 DNA to super...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed