Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM50068664'
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(CHEMBL191751 | 2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-...)
Affinity DataKi:  0.308nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(CHEMBL191751 | 2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-...)
Affinity DataKi:  0.308nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50068664(CHEMBL191751 | 2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(CHEMBL191751 | 2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(CHEMBL191751 | 2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-...)
Affinity DataKi:  1.22nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50068664(CHEMBL191751 | 2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-...)
Affinity DataKi:  6.10nMAssay Description:Affinity towards human Opioid receptor delta 1 on CHO cell membranes using [3H]DPDPE displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed