Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Endoplasmic reticulum chaperone BiP' and Ligand = 'BDBM31712'
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31712BDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31712BDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31712BDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31712BDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed