Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Endothelin-1 receptor' and Ligand = 'BDBM25761'
TargetEndothelin-1 receptor(Human)
Janssen Pharmaceutica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataIC50: 5.01E+3nMAssay Description:Antagonist activity at human wild-type ETA receptor expressed in CHO-K1 cells assessed as endothelin-1-induced calcium by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Janssen Pharmaceutica

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type ETA receptor expressed in CHO-K1 cells assessed as calcium level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed