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Found 5 Enz. Inhib. hit(s) with Target = 'Ephrin type-A receptor 3' and Ligand = 'BDBM13533'
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50: <1.00E+3nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of EPHA3More data for this Ligand-Target Pair
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd:  580nMAssay Description:Average Binding Constant for EPHA3; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd:  880nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd:  880nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair