Found 26 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM19459' 
Affinity DataKi: 370nMAssay Description:Inhibition of binding of 17 beta-estradiol to human Estrogen receptor alphaMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 9.70nMAssay Description:Inhibition of human LBD of of ERalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 29.4nMAssay Description:Displacement of [3H]17beta-estradiol from recombinant human ERalpha expressed in 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Binding affinity against human estrogen receptor alpha in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Displacement of [3H]estradiol from human recombinant ERalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Binding affinity for human Estrogen receptor alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Binding affinity towards human estrogen receptor alpha(ERalpha)More data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Binding affinity for human Estrogen receptor alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Inhibitory concentration against human ER alpha expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Displacement of [3H]17beta-estradiol from recombinant human ERalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of binding of 17 beta-estradiol to human Estrogen receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+3nM EC50: 956nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
Affinity DataIC50: 2.15E+3nMAssay Description:Binding affinity to human ERalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.92E+3nM EC50: 48nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assay was performed by using 96-well microtiterplates containing ER, 17beta-estradiol, and the test compound to be tested and SPA...More data for this Ligand-Target Pair
Affinity DataIC50: 4.66E+3nMAssay Description:Binding affinity for human Estrogen receptor AlphaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.66E+3nMAssay Description:Binding affinity for human Estrogen receptor AlphaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.68E+3nMAssay Description:The binding affinity and selectivity of candidate molecules yielded from
database screening were determined by a fluorescent polarization
competiti...More data for this Ligand-Target Pair
Affinity DataIC50: 4.74E+3nMAssay Description:Displacement of EL red from human full-length ER-alpha expressed in baculovirus expression system incubated for 2 hrs by fluorescence polarization as...More data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Binding affinity towards estrogen receptor alpha by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
Affinity DataEC50: 950nMAssay Description:Ability to activate estrogen receptor 1-mediated transcription.More data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Estrogenic activity at ERalpha in human Ishikawa cells assessed as induction of alkaline phosphatase activity using p-nitrophenol as substrate treate...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 810nMAssay Description:Agonist activity at human ERalpha expressed in yeast AH109 by yeast two hybrid assayMore data for this Ligand-Target Pair
