Affinity DataKi: 249nMAssay Description:Displacement of (R,S)-[5-methyl-3H]AMPA from rat recombinant flop iGluR3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity to full length rat GluA3More data for this Ligand-Target Pair
Affinity DataKi: 7.40E+3nMAssay Description:Binding affinity to rat GluA3-LBD (GluK3-S1S2)More data for this Ligand-Target Pair
Affinity DataEC50: 2.34E+4nMAssay Description:Agonist activity at GluA3 receptor (unknown origin) expressed in HEK293 cells assessed induction of S-glutamate-induced calcium flux measured after 9...More data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+4nMAssay Description:Agonist activity at rat recombinant GluR3 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assa...Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 6.70E+4nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Activity at rat cloned iGluR3 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+4nMAssay Description:Agonist activity at rat recombinant GluA3 receptor flip isoform expressed in HEK293 cells assessed as effect on cyclothiazide-induced calcium flux by...More data for this Ligand-Target Pair
Affinity DataEC50: 3.66E+3nMAssay Description:Agonist activity at recombinant GluA3 receptor flop isoform expressed in Xenopus oocytes co-expressing gamma2-TARPMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+4nMAssay Description:Agonist activity at GluA3 receptor (unknown origin) expressed in HEK293 cells assessed induction of S-glutamate-induced calcium flux measured after 9...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at rat recombinant GluA3 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.12E+4nMAssay Description:Agonist activity at recombinant rat GluA3 receptor flip isoform expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+4nMAssay Description:Agonist activity at recombinant GluA3 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair