Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 3' and Ligand = 'BDBM50069111'
TargetGlutamate receptor ionotropic, kainate 3(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069111BDBM50069111((2S,4S)-2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioi...)
Affinity DataIC50: 380nMAssay Description:Binding affinity against Ionotropic glutamate receptor using ACPD sensitive [3H]- glutamate displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069111BDBM50069111((2S,4S)-2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioi...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity against Ionotropic glutamate receptor using [3H]- CGS-19755 displacement from rat forebrain preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed