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Found 2 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50517283'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]-His9 ghrelin from SNAP-tagged human GHSR expressed in HEK293T cells after 3 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataEC50:  1.5nMAssay Description:Inverse agonist activity at SNAP-tagged human GHSR expressed in HEK293T cells assessed as reduction in inositol phosphate production after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed