Found 12 Enz. Inhib. hit(s) with Target = 'Heat shock protein HSP 90-alpha' and Ligand = 'BDBM50008057'
Affinity DataKi: 29nMAssay Description:Inhibition of FITC-GA binding to Hsp90alpha (unknown origin) ATPase site after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human N terminal his-tagged HSP90 alpha (1 to 732 residues) expressed in Escherichia coli measured after 60 mins by Floures...More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of FITC-labeled geldanamycin binding to human Hsp90alpha by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of GA-FITC binding to human recombinant Hsp90alpha incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 309nMAssay Description:Inhibition of FITC-GA binding to N-terminal domain of HSP90alpha (unknown origin) after 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Displacement of GA-FITC from human recombinant HSP90alpha ATP-binding site by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Inhibition of HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 assessed as reduction in ATPase activity in presence of PEP, NADH and A...More data for this Ligand-Target Pair
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of human HSP90alpha expressed in yeast assessed as growth inhibition of host after 72 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.83E+4nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human full-length C-terminal His-tagged HSP90alpha expressed in Escherichia coli after 3 hrs b...More data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding affinity to recombinant HSP90-alpha (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 388nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 900nMAssay Description:Binding affinity to HSP90-alpha (unknown origin) expressed in Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair