Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Heparanase' and Ligand = 'BDBM50165652'
TargetHeparanase(Human)
Sharif University of Technology

Curated by ChEMBL
LigandPNGBDBM50165652(2-(2-(4-(3-(4-bromophenyl)acrylamido)-3-fluorophen...)
Affinity DataIC50: 398nMAssay Description:Inhibition of heparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHeparanase(Human)
Sharif University of Technology

Curated by ChEMBL
LigandPNGBDBM50165652(2-(2-(4-(3-(4-bromophenyl)acrylamido)-3-fluorophen...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Sharif University of Technology

Curated by ChEMBL
LigandPNGBDBM50165652(2-(2-(4-(3-(4-bromophenyl)acrylamido)-3-fluorophen...)
Affinity DataIC50: 400nMAssay Description:Inhibition of human heparanase assessed as reduction in basic fibroblast growth factor binding incubated for 2 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHeparanase(Human)
Sharif University of Technology

Curated by ChEMBL
LigandPNGBDBM50165652(2-(2-(4-(3-(4-bromophenyl)acrylamido)-3-fluorophen...)
Affinity DataIC50: 7.68E+3nMAssay Description:Recombinant human active heparanase derived from Chinese hamster ovary cells was from R&D Systems. Bovine serum albumin-coated 96 well microplates (9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2023
Entry Details
US Patent