Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50138119'
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences

Curated by ChEMBL
LigandPNGBDBM50138119(CHEMBL3753475)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences

Curated by ChEMBL
LigandPNGBDBM50138119(CHEMBL3753475)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences

Curated by ChEMBL
LigandPNGBDBM50138119(CHEMBL3753475)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed on CHO-K1 cells assessed as cAMP level by luciferase gene reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed