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Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50222968'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50222968(Cipralisant | GT-2331)
Affinity DataKi:  0.126nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50222968(Cipralisant | GT-2331)
Affinity DataKi:  0.195nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222968(Cipralisant | GT-2331)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed