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Found 4 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50458224'
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL
LigandPNGBDBM50458224(CHEMBL2297871)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]iodoproxyfan from human H3R expressed in CHOK1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Medical University

Curated by ChEMBL
LigandPNGBDBM50458224(CHEMBL2297871)
Affinity DataKi:  4nMAssay Description:Binding affinity to Rattus norvegicus (rat) H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL
LigandPNGBDBM50458224(CHEMBL2297871)
Affinity DataKi:  11nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL
LigandPNGBDBM50458224(CHEMBL2297871)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human H3R expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed