Found 4 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300' and Ligand = 'BDBM188519' 
Affinity DataIC50: 67nMAssay Description:Inhibition of EP300 bromodomain (unknown origin) incubated for 20 mins by AlphaLISA methodMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 230nMAssay Description:Inhibition of biotinylated-H4KAc4 binding to human His6-tagged EP300 (A1040 to G1161 residues) expressed in Escherichia coli BL21(DE3) after 2.5 hrs ...More data for this Ligand-Target Pair
Affinity DataKd: 3.18E+7nMAssay Description:Inhibition of human BRD4 BD1 (67 to 152 residues) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra...More data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Binding affinity to human p300 by ITC analysisMore data for this Ligand-Target Pair
