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Found 1 Enz. Inhib. hit(s) with Target = 'Histone-arginine methyltransferase CARM1' and Ligand = 'BDBM27643'
TargetHistone-arginine methyltransferase CARM1(Mus musculus (mouse))
Methylgene

LigandPNGBDBM27643(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...)
Affinity DataIC50:  300nMpH: 9.0 T: 2°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed